Compile Data Set for Download or QSAR
Found 21 of Enz. Inhib. data with enzyme = 'Nociceptin receptor' and Substrate = 'BDBM26957'
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26976(2-benzoylquinazoline analogue, (1R, 2S)-17 | N-(4-...)copy SMILEScopy InChI
Affinity DataKi:  1.40nM ΔG°:  -12.1kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26975(2-benzoylquinazoline analogue, (rac)-17 | N-{4-[(2...)copy SMILEScopy InChI
Affinity DataKi:  2.10nM ΔG°:  -11.8kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26973((1R,2S)-2-({2-[(E)-2-(4-chlorophenyl)ethenyl]-6-me...)copy SMILEScopy InChI
Affinity DataKi:  43nM ΔG°:  -10.0kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26971(3-[6-({2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylq...)copy SMILEScopy InChI
Affinity DataKi:  89nM ΔG°:  -9.61kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26956(N-(6-aminohexyl)-2-[(E)-2-(4-chlorophenyl)ethenyl]...)copy SMILEScopy InChI
Affinity DataKi:  133nM ΔG°:  -9.37kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26977(2-benzoylquinazoline analogue, (1S, 2R)-17 | N-(4-...)copy SMILEScopy InChI
Affinity DataKi:  140nM ΔG°:  -9.34kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26974(4-({2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylquin...)copy SMILEScopy InChI
Affinity DataKi:  152nM ΔG°:  -9.29kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26972(3-[4-({2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylq...)copy SMILEScopy InChI
Affinity DataKi:  160nM ΔG°:  -9.26kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26969(1-N-{2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylqui...)copy SMILEScopy InChI
Affinity DataKi:  162nM ΔG°:  -9.26kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26965(4-aminoquinazoline derivative, 7h | N-(4-aminobuty...)copy SMILEScopy InChI
Affinity DataKi:  194nM ΔG°:  -9.15kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26968((1S,2R)-1-N-{2-[(E)-2-(4-chlorophenyl)ethenyl]-6-m...)copy SMILEScopy InChI
Affinity DataKi:  200nM ΔG°:  -9.13kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26960(4-aminoquinazoline derivative, 7c | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  232nM ΔG°:  -9.04kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26963(4-aminoquinazoline derivative, 7f | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  292nM ΔG°:  -8.91kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26964(4-aminoquinazoline derivative, 7g | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  294nM ΔG°:  -8.90kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26958(4-aminoquinazoline derivative, 7a | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  383nM ΔG°:  -8.75kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26961(4-aminoquinazoline derivative, 7d | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  420nM ΔG°:  -8.69kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26967((1S,2S)-1-N-{2-[(E)-2-(4-chlorophenyl)ethenyl]-6-m...)copy SMILEScopy InChI
Affinity DataKi:  538nM ΔG°:  -8.55kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26962(4-aminoquinazoline derivative, 7e | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  653nM ΔG°:  -8.43kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26970(1-N-{2-[(E)-2-(4-chlorophenyl)ethenyl]-6-methylqui...)copy SMILEScopy InChI
Affinity DataKi:  795nM ΔG°:  -8.32kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26959(4-aminoquinazoline derivative, 7b | N-(6-aminohexy...)copy SMILEScopy InChI
Affinity DataKi:  808nM ΔG°:  -8.31kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Nippon Shinyaku Co.

LigandPNGBDBM26966(4-aminoquinazoline derivative, 7i | N-(2-aminoethy...)copy SMILEScopy InChI
Affinity DataKi:  972nM ΔG°:  -8.20kcal/molepH: 7.8 T: 2°CAssay Description:Competitive binding displacement analysis was performed with membranes prepared from CHO-K1 cells stably expressing receptors. After incubation, samp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52MX5PubMed